EDNRA

EDNRA

EDNRA Overview

Molecule Name
Endothelin receptor type A
Synonyms
endothelin receptor type A, ETA,ET-A,ETAR,ETRA,MFDA,ETA-R,hET-AR
Drug Development Progress
Drugs in Clinical Trials11
Approved Drugs8
Highest Development StageApproved
Target Synonym
Endothelin Receptor Type A,EDNRA,ETA-R,Endothelin-1 receptor,hET-AR,ETRA,ET-A,ETA,Endothelin-1-Specific Receptor,Endothelin Receptor Subtype A,G Protein-Coupled Receptor,ETAR,MFDA,Receptor, Endothelin A
Background
EDNRA encodes the endothelin type A receptor, a G protein-coupled receptor mediating vasoconstriction and cell proliferation upon endothelin-1 binding. Overexpression contributes to pulmonary arterial hypertension, cardiovascular disorders, and cancer progression. Selective EDNRA antagonists offer therapeutic potential for managing hypertension, fibrosis, and tumor angiogenesis.

EDNRA Product List

Species
  • Human(3)
Tag
  • -(2)
  • His Tag & Flag Tag(1)
Host
  • HEK293(2)
  • E. coli(1)
Conjugate
  • Unconjugated(2)
  • Biotin-labeled(1)
Grade
  • RUO(3)
Low Endotoxin
  • No(3)
MoleculeCat. No.Product NameSpeciesHostStructurePurityActivitySize&PriceAdd to Cart
EDNRA
Human EDNRA Full Length Protein, His,Flag Tag (Detergent)
Human
E. coli
SDS-PAGE
ELISA

$496.00

20ug
EDNRA
Human EDNRA Full Length Protein (VLP)
Human
HEK293
ELISAIdentity

$620.00

20ug
EDNRA
Biotinylated Human EDNRA Full Length Protein (VLP)
Human
HEK293
ELISAIdentity

$620.00

20ug
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Clinical Drug Information

English NameResearch CodeHighest Development StageCompanyIndicationClinical Trial
SC-0062SC-0062; WX-013Phase 3 ClinicalShijiazhuang Zhikang Hongren New Drug Development Co Ltd
Altitude Sickness; Diabetic Nephropathies; Glomerulonephritis, IGA; Kidney Diseases; Pulmonary Arterial Hypertension
Details
Zibotentan/DapagliflozinPhase 3 ClinicalAstrazeneca Ab, AstraZeneca global R & D (China) Co Ltd
Albuminuria; Kidney Diseases; Renal Insufficiency, Chronic
Details
PatecibartGMA-301; GMA-301-A; GMA-301-BPhase 2 ClinicalGmax Biopharm Llc
Pulmonary Arterial Hypertension
Details
ZibotentanZD-4054; AZD-4054Phase 2 ClinicalAstrazeneca Plc
Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Hepatic Insufficiency; Hypertension, Portal; Intermittent Claudication; Liver Cirrhosis; Lung Neoplasms; Metastatic breast cancer; Microvascular Angina; Neoplasm Metastasis; Ovarian Neoplasms; Peripheral Arterial Disease; Prostatic Neoplasms; Renal Insufficiency; Renal Insufficiency, Chronic; Scleroderma, Limited; Scleroderma, Systemic; Solid tumours
Details
SAL-0120SAL-0120; SAL0120Phase 2 ClinicalShenzhen Salubris Pharmaceuticals Co Ltd
Essential Hypertension; Glomerulonephritis, IGA; Hypertension; Renal Insufficiency, Chronic
Details
HS-10390HS-10390; HS10390Phase 2 ClinicalChangzhou Hengbang Pharmaceutical Co Ltd, Shanghai Hansoh Biomedical Co Ltd
Glomerulonephritis, IGA; Glomerulosclerosis, Focal Segmental; Renal Insufficiency, Chronic
Details
BQ-123CGS-26343; BQ-123; PMZ-2123Phase 1 ClinicalMidwestern University
Cardiovascular Diseases; Coronary Artery Disease; Diabetic Ketoacidosis; Heart Failure; Hypertension; Hypertension, Pulmonary; Hypoxia, Brain; Metabolic Syndrome; Multiple System Atrophy; Pain; Proteinuria; Pure Autonomic Failure; Renal Insufficiency, Chronic; ST Elevation Myocardial Infarction
Details
GMA-131GMA-131Phase 1 ClinicalGmax Biopharm Llc, Gmaxx Biologics Ltd
Diabetic Nephropathies
Details
AK-1960AK1960; AK-1960Phase 1 Clinical
Renal Insufficiency, Chronic
Details
GLX-002GLX-002; GLX002Phase 1 ClinicalYabao Pharmaceutical Co Ltd Beijing
Pulmonary Arterial Hypertension
Details
Bosentan Orally Disintegrating Tablets(Beijing Sunho Pharma)Phase 1 ClinicalBeijing Sunho Pharmaceutical Co Ltd
Pulmonary Arterial Hypertension
Details

Marketed Drug Information

English NameResearch CodeHighest Development StageCompanyFirst Brand NameFirst Approved CountryFirst IndicationFirst Approved CompanyFirst Approved DateIndicationClinical Trial
Clazosentan SodiumRo-61-1790; ACT-108475; AXV-034; VML-588; AXV-034343ApprovedF. Hoffmann-La Roche LtdPivlazJapanSubarachnoid Hemorrhage; Brain Ischemia; Vasospasm, Intracranial; Cerebral InfarctionIdorsia Pharmaceuticals Ltd2022-01-20
Aneurysm; Brain Ischemia; Cerebral Infarction; Subarachnoid Hemorrhage; Vasospasm, Intracranial
Details
Macitentan/TadalafilApprovedActelion Pharmaceuticals LtdOPSYNVI, YuvanciUnited StatesPulmonary Arterial HypertensionActelion Pharmaceuticals Us Inc2024-03-22
Phenylketonurias; Pulmonary Arterial Hypertension
Details
AmbrisentanLU-208075; BSF-208075; GSK-132576AApprovedAbbott LaboratoriesLetairis, Volibris, 凡瑞克United StatesPulmonary Arterial HypertensionGilead Sciences Inc2007-06-15
Acute Kidney Injury; Anemia, Sickle Cell; Ascites; Coronavirus Disease 2019 (COVID-19); Hepatorenal Syndrome; Hypertension; Hypertension, Portal; Hypertension, Pulmonary; Hypoxia; Idiopathic Pulmonary Fibrosis; Liver Cirrhosis; Pulmonary Arterial Hypertension; Sarcoidosis; Scleroderma, Systemic; Thromboembolism; Vascular Diseases
Details
SparsentanPS-433540; BMS-346567; RE-021ApprovedBristol-Myers Squibb CompanyFilspariUnited StatesGlomerulonephritis, IGATravere Therapeutics Inc2023-02-17
Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Autoimmune Diseases; Cardiovascular Diseases; Glomerulonephritis; Glomerulonephritis, IGA; Glomerulosclerosis, Focal Segmental; Hypertension; Immune System Diseases; Kidney Diseases; Nephritis, Hereditary; Nephrosis, Lipoid; Proteinuria; Purpura, Schoenlein-Henoch
Details
Bosentan HydrateACT-050088; HGP-1206; Ro-47-0203; Ro-47-0203/029; Ro-47-0203/039ApprovedF. Hoffmann-La Roche LtdStayveer, 全可利, TracleerUnited StatesPulmonary Arterial HypertensionActelion Pharmaceuticals Ltd2001-11-20
Anemia, Sickle Cell; Chronic thromboembolic pulmonary hypertension; Coronary Vasospasm; Diabetes Mellitus; Diabetes Mellitus, Type 2; Fibrosis; Giant Cell Arteritis; Glaucoma; Heart Defects, Congenital; Heart Septal Defects, Atrial; Hepatopulmonary Syndrome; Hypertension; Hypertension, Pulmonary; Idiopathic Pulmonary Fibrosis; Liver Cirrhosis; Lung Diseases, Interstitial; Persistent Fetal Circulation Syndrome; Pulmonary Arterial Hypertension; Pulmonary Fibrosis; Sarcoidosis; Scleroderma, Systemic; Sleep Apnea Syndromes; Takayasu Arteritis; Ulcer; Vasculitis
Details
MacitentanACT-064992; Actelion-1; JNJ-67896062ApprovedActelion Pharmaceuticals LtdZependo, Opsumit, 傲朴舒United StatesPulmonary Arterial HypertensionActelion Pharmaceuticals Us Inc2013-10-18
Anemia, Sickle Cell; Angina Pectoris; Chronic Disease; Chronic thromboembolic pulmonary hypertension; Eisenmenger Complex; Glioblastoma; Heart Defects, Congenital; Heart Failure; Heart Failure, Diastolic; Hypertension, Pulmonary; Idiopathic Pulmonary Fibrosis; Pulmonary Arterial Hypertension; Pulmonary Embolism; Scleroderma, Systemic; Scleroderma-associated interstitial lung diseases; Thromboembolism; Ulcer
Details
AprocitentanACT-132577; AC-080; JNJ-2820ApprovedActelion Pharmaceuticals Ltd, Idorsia Pharmaceuticals LtdTRYVIO, JERAYGOUnited StatesHypertensionIdorsia Pharmaceuticals Ltd2024-03-19
Essential Hypertension; Hepatic Insufficiency; Hypertension; Renal Insufficiency, Chronic
Details
Atrasentan hydrochlorideABT-147627; (+)-A-127722; Abbott-147627; A-147627; ABT-627; A-1476271; CHK-01; EXV 811ApprovedAbbvie IncVanrafia, 诺锐达, XinlayUnited StatesGlomerulonephritis, IGA; ProteinuriaNovartis Pharmaceutical Corp, Novartis Pharma Ag2025-04-02
Abdominal Neoplasms; Adenocarcinoma; CNS Embryonal Tumor; Diabetes Mellitus; Diabetic Nephropathies; Fallopian Tube Neoplasms; Glomerulonephritis, IGA; Glomerulosclerosis, Focal Segmental; Kidney Diseases; Kidney Neoplasms; Neoplasm Metastasis; Nephritis, Hereditary; Ovarian Neoplasms; Prostatic Neoplasms; Proteinuria; Renal Insufficiency, Chronic; Vascular Diseases
Details
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